Access to chiral phthalidyl ester prodrugs via an isothiourea-catalyzed dynamic kinetic resolution reaction
- 25 March 2025
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Organic & Biomolecular Chemistry
- Vol. 23 (15) , 3680-3688
Abstract
An isothiourea-catalyzed acylative dynamic kinetic resolution reaction has been developed for the synthesis of chiral phthalidyl ester prodrugs.Keywords
Funding Information
- National Natural Science Foundation of China (22371058)
- National Natural Science Foundation of China (U23A20201)
- National Natural Science Foundation of China (22071036)
- National Basic Research Program of China (2022YFD1700300)
- Guizhou University ((2023)29)
- Guizhou Provincial Science and Technology Department (Qiankehejichu-ZK[2024]Key009)
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