Synthesis of 1-(6-chloro-1,1-dioxo-1,4,2-benzodithiazin-3-yl)semi-carbazides and their transformation into 4-chloro-2-mercapto-N-(4,5-dihydro-5-oxo-4-phenyl-1H-1,2,4-triazol-3-yl)benzenesulfonamides as potential anticancer and anti-HIV agents
- 30 June 2003
- journal article
- Published by Elsevier in Il Farmaco
- Vol. 58 (6) , 423-429
Abstract
No abstract availableKeywords
This publication has 16 references indexed in Scilit:
- Synthesis and Antiviral Activity of New Anti-HIV Amprenavir BioisosteresJournal of Medicinal Chemistry, 2002
- Carbonic Anhydrase Inhibitors. A General Approach for the Preparation of Water-Soluble Sulfonamides Incorporating Polyamino−Polycarboxylate Tails and of Their Metal Complexes Possessing Long-Lasting, Topical Intraocular Pressure-Lowering PropertiesJournal of Medicinal Chemistry, 2002
- Phenoxyphenyl SulfoneN-Formylhydroxylamines (Retrohydroxamates) as Potent, Selective, Orally Bioavailable Matrix Metalloproteinase InhibitorsJournal of Medicinal Chemistry, 2001
- A New Type of Mixed Anhydride and Its Applications to the Synthesis of 7-Substituted 8-Chloro-5,5-dioxoimidazo[1,2-b][1,4,2]benzodithiazines with in Vitro Antitumor ActivityJournal of Medicinal Chemistry, 2001
- Synthesis and anti-HIV activity of 4-[(1,2-dihydro-2-oxo-3H-indol-3-ylidene) amino]-N(4,6-dimethyl-2-pyrimidinyl)-benzene sulfonamide and its derivativesEuropean Journal of Pharmaceutical Sciences, 2001
- Synthesis and in vitro anticancer and anti-HIV evaluation of new 2-mercaptobenzenesulfonamidesIl Farmaco, 2001
- Potent and Selective Carboxylic Acid-Based Inhibitors of Matrix MetalloproteinasesJournal of Medicinal Chemistry, 2001
- A Facile Synthesis and Chemical Properties of 3,4-Dihydro-2H-1,5,2-benzo[f]dithiazepin-3-ones with Potential Anticancer ActivityHETEROCYCLES, 2001
- 2-Mercaptobenzenesulphonamides as Novel Inhibitors of Human Immunodeficiency virus Type 1 Integrase and ReplicationAntiviral Chemistry and Chemotherapy, 1997
- Design and discovery of HIV-1 integrase inhibitorsDrug Discovery Today, 1997