Active site mapping of trypsin, thrombin and matriptase-2 by sulfamoyl benzamidines
Authors:
- Marit StirnbergMSMarit Stirnberg
- Verena LülsdorffVLVerena Lülsdorff
- Daniela HäußlerDHDaniela Häußler
- Eva MaurerEMEva Maurer
- Michael GütschowMGMichael Gütschow
- 1 November 2012
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry
- Vol. 20 (21) , 6489-6505
Abstract
No abstract availableKeywords
This publication has 76 references indexed in Scilit:
- Synthesis and Antiprotozoal Activity of Pyridyl Analogues of PentamidineJournal of Medicinal Chemistry, 2009
- Synthesis and in Vitro Antiprotozoal Activities of Dicationic 3,5-DiphenylisoxazolesJournal of Medicinal Chemistry, 2007
- Identification of the Missing Component in the Mitochondrial Benzamidoxime Prodrug-converting System as a Novel Molybdenum EnzymeJournal of Biological Chemistry, 2006
- Piperazine-linked bisbenzamidines: a novel class of antileishmanial agentsEuropean Journal of Medicinal Chemistry, 2004
- Parallel Solution-Phase Synthesis of Conformationally Restricted Congeners of Pentamidine and Evaluation of Their Antiplasmodial ActivitiesJournal of Medicinal Chemistry, 2004
- Lessons Learned from Marketed and Investigational ProdrugsJournal of Medicinal Chemistry, 2004
- Sulfonyl-phenyl-ureido benzamidinesBioorganic & Medicinal Chemistry Letters, 2004
- Design of Selective Thrombin Inhibitors Based on the (R)-Phe-Pro-Arg SequenceJournal of Medicinal Chemistry, 2002
- REDUCTION OFN-HYDROXYLATED COMPOUNDS: AMIDOXIMES (N-HYDROXYAMIDINES) AS PRO-DRUGS OF AMIDINESDrug Metabolism Reviews, 2002
- The Chemistry of Imidates.Chemical Reviews, 1961