Silver mediated direct C–H arylation of 3-bromoisothiazole-5-carbonitrile

This publication has 47 references indexed in Scilit:

• Discovery of (1R,2R)-N-(4-(6-isopropylpyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide, a potent and orally efficacious mGlu5 receptor negative allosteric modulator
  Bioorganic & Medicinal Chemistry Letters, 2013
• Synthetic Inhibitors of the Fungal Detoxifying Enzyme Brassinin Oxidase Based on the Phytoalexin Camalexin Scaffold
  Journal of Agricultural and Food Chemistry, 2009
• Diaryl-dithiolanes and -isothiazoles: COX-1/COX-2 and 5-LOX-inhibitory, OH scavenging and anti-adhesive activities
  Bioorganic & Medicinal Chemistry, 2009
• Synthesis and pharmacology of glutamate receptor ligands: new isothiazole analogues of ibotenic acid
  Organic & Biomolecular Chemistry, 2006
• 3-(Indol-2-yl)indazoles as Chek1 kinase inhibitors: Optimization of potency and selectivity via substitution at C6
  Bioorganic & Medicinal Chemistry Letters, 2006
• Discovery of 3-hydroxy-4-carboxyalkylamidino-5-arylamino-isothiazoles as potent MEK1 inhibitors
  Bioorganic & Medicinal Chemistry Letters, 2006
• Design, synthesis, and antifungal activity of inhibitors of brassilexin detoxification in the plant pathogenic fungus Leptosphaeria maculans
  Bioorganic & Medicinal Chemistry, 2006
• The chemistry of isothiazoles
  Tetrahedron, 2003
• Regiospecific Suzuki coupling of 3,5-dichloroisothiazole-4-carbonitrile
  Organic & Biomolecular Chemistry, 2003
• Isothiazoles (1,2-thiazoles): synthesis, properties and applications
  Russian Chemical Reviews, 2002