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  2. Publications
  3. Bioavailable dual-protein degraders of CK1α and transcriptional kinase CDK9 as potential therapeutics for hematological malignancies
  1. Home
  2. Publications
  3. Bioavailable dual-protein degraders of CK1α and transcriptional kinase CDK9 as potential therapeutics for hematological malignancies

Bioavailable dual-protein degraders of CK1α and transcriptional kinase CDK9 as potential therapeutics for hematological malignancies

Authors:
  • Imelda Calderon
    Imelda Calderon
  • Robert Sullivan
    Robert Sullivan
  • Leah Fung
    Leah Fung
  • Aparajita Chourasia
    Aparajita Chourasia
  • Frank Mercurio
    Frank Mercurio
  • BMBrooke McElwee
    Brooke McElwee
  • Yinon Ben-Neriah
    Yinon Ben-Neriah
  • ETEduardo Torres
    Eduardo Torres
  • Paul Erdman
    Paul Erdman
  • Kyle Chan
    Kyle Chan
  • David Hecht
    David Hecht

Open Access
Publisher website
Google Scholar
  • 30 November 2020
    • conference paper
    • Published by American Chemical Society (ACS)
    • DOI:10.1021/scimeetings.0c07406
Abstract
No abstract available
Keywords
  • RECEIVED FDA
  • FDA APPROVAL
  • IND APPLICATION
  • BIOAVAILABLE DUAL-PROTEIN
  • MYELOID LEUKEMIA
  • DUAL-PROTEIN DEGRADERS
  • POTENTIAL THERAPEUTICS
  • HEMATOLOGICAL MALIGNANCIES
  • MALIGNANCIES BIOTHERYX
  • DITOSYLATED SALT
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