Construction of a spiro[pyrazolone-4,2′-pyridoindole] scaffold via a [3 + 3] cycloaddition of 2-indolylmethanol with a 4-aminopyrazolone-derived azomethine ylide
- 9 September 2021
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Organic & Biomolecular Chemistry
- Vol. 19 (39) , 8530-8538
Abstract
A one-pot [3 + 3] cycloaddition of 2-indolylmethanol with an in situ generated azomethine ylide derived from 4-aminopyrazolone is developed to access the spiro[pyrazolone–pyridoindole] scaffold.Keywords
Funding Information
- Central University Basic Research Fund of China (DUT21LAB134)
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