Simple and facile synthesis of tetralone-spiro-glutarimides and spiro-bisglutarimides from Baylis–Hillman acetates
- 6 February 2008
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Organic & Biomolecular Chemistry
- Vol. 6 (6) , 1034-1039
Abstract
A simple and convenient synthesis of di(E)-arylidene-tetralone-spiro-glutarimides from Baylis–Hillman acetates via an interesting biscyclization strategy involving facile C–C and C–N bond formation is described. Also, one-pot multistep transformation of the Baylis–Hillman acetates into di(E)-arylidene-spiro-bisglutarimides is presented.Keywords
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