Danazol oral absorption modelling in the fasted dog: An example of mechanistic understanding of formulation effects on drug pharmacokinetics
- 1 August 2019
- journal article
- research article
- Published by Elsevier in European Journal of Pharmaceutics and Biopharmaceutics
- Vol. 141, 191-209
Abstract
No abstract availableKeywords
This publication has 40 references indexed in Scilit:
- Evaluation of a Nanoemulsion Formulation Strategy for Oral Bioavailability Enhancement of Danazol in Rats and DogsJournal of Pharmaceutical Sciences, 2013
- Excipient-Mediated Supersaturation Stabilization in Human Intestinal FluidsMolecular Pharmaceutics, 2011
- Sodium/glucose cotransporter-1, sweet receptor, and disaccharidase expression in the intestine of the domestic dog and cat: two species of different dietary habitAmerican Journal of Physiology-Regulatory, Integrative and Comparative Physiology, 2011
- Drug Supersaturation in Simulated Human Intestinal Fluids Representing Different Nutritional StatesJournal of Pharmaceutical Sciences, 2010
- Identification of Novel Substrates for Human Cytochrome P450 2J2Drug Metabolism and Disposition, 2010
- Population-Based Mechanistic Prediction of Oral Drug AbsorptionThe AAPS Journal, 2009
- Estimation of effective intestinal membrane permeability considering bile micelle solubilisationInternational Journal of Pharmaceutics, 2009
- Comparison of a Miniaturized Shake-Flask Solubility Method with Automated Potentiometric Acid/Base Titrations and Calculated SolubilitiesJournal of Pharmaceutical Sciences, 2005
- Effect of simulated intestinal fluid on drug permeability estimation across Caco-2 monolayersInternational Journal of Pharmaceutics, 2004
- Pharmaceutical Applications of Cyclodextrins. 2. In Vivo Drug DeliveryJournal of Pharmaceutical Sciences, 1996