Sustained Activation of a G Protein-coupled Receptor via “Anchored” Agonist Binding
Authors:
- Andrew P. SpasoffASAndrew P. Spasoff
- Robert A. ColemanRCRobert A. Coleman
- Malcolm JohnsonMJMalcolm Johnson
- Stephen B. LiggettSLStephen B. Liggett
Open Access
- 1 September 1996
- journal article
- Published by Elsevier in Journal of Biological Chemistry
- Vol. 271 (39) , 24029-24035
Abstract
No abstract availableKeywords
This publication has 22 references indexed in Scilit:
- SalmeterolMedicinal Research Reviews, 1995
- Why are long-acting beta-adrenoceptor agonists long-acting?European Respiratory Journal, 1994
- Modeling of transmembrane seven helix bundlesProtein Engineering, Design and Selection, 1993
- A Comparison of Salmeterol with Albuterol in the Treatment of Mild-to-Moderate AsthmaNew England Journal of Medicine, 1992
- The 1990 Lilly Prize Lecture. A way of looking at agonism and antagonism: lessons from salbutamol, salmeterol and other beta‐ adrenoceptor agonists.British Journal of Clinical Pharmacology, 1991
- Model for the structure of bacteriorhodopsin based on high-resolution electron cryo-microscopyJournal of Molecular Biology, 1990
- WHAT IF: A molecular modeling and drug design programJournal of Molecular Graphics, 1990
- [71] Use of eukaryotic expression technology in the functional analysis of cloned genes1987
- Measurement of protein using bicinchoninic acidAnalytical Biochemistry, 1985
- Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionBiochemical Pharmacology, 1973