Structural and biochemical studies of the PDGFRA kinase domain
- 1 September 2016
- journal article
- Published by Elsevier in Biochemical and Biophysical Research Communications
- Vol. 477 (4) , 667-672
Abstract
No abstract availableKeywords
Funding Information
- National Key Research and Development Program of China (2012CB917202)
- National Natural Science Foundation of China (31270769)
- Ministry of Education of the People's Republic of China (NCET-12-0013)
This publication has 26 references indexed in Scilit:
- PHENIX: a comprehensive Python-based system for macromolecular structure solutionActa Crystallographica Section D Structural Biology, 2010
- Novel mutant-selective EGFR kinase inhibitors against EGFR T790MNature, 2009
- KIT kinase mutants show unique mechanisms of drug resistance to imatinib and sunitinib in gastrointestinal stromal tumor patientsProceedings of the National Academy of Sciences, 2009
- Phasercrystallographic softwareJournal of Applied Crystallography, 2007
- Structures of Lung Cancer-Derived EGFR Mutants and Inhibitor Complexes: Mechanism of Activation and Insights into Differential Inhibitor SensitivityCancer Cell, 2007
- FMS receptor for M-CSF (CSF-1) is sensitive to the kinase inhibitor imatinib and mutation of Asp-802 to Val confers resistanceOncogene, 2005
- PDGFRA Mutations in Gastrointestinal Stromal Tumors: Frequency, Spectrum and In Vitro Sensitivity to ImatinibJournal of Clinical Oncology, 2005
- Coot: model-building tools for molecular graphicsActa Crystallographica Section D Structural Biology, 2004
- The Structural Basis for Autoinhibition of FLT3 by the Juxtamembrane DomainMolecular Cell, 2004
- Src Family Kinases Negatively Regulate Platelet-derived Growth Factor α Receptor-dependent Signaling and Disease ProgressionJournal of Biological Chemistry, 2000