Determination of permeability and lipophilicity of pyrazolo-pyrimidine tyrosine kinase inhibitors and correlation with biological data

This publication has 31 references indexed in Scilit:

• Correlation between PAMPA permeability and cellular activities of hepatitis C virus protease inhibitors
  Biochemical Pharmacology, 2008
• Identification of a Novel Pyrazolo[3,4-d]pyrimidine Able To Inhibit Cell Proliferation of a Human Osteogenic Sarcoma in Vitro and in a Xenograft Model in Mice
  Journal of Medicinal Chemistry, 2007
• Molecular Lipophilicity in Protein Modeling and Drug Design
  Current Medicinal Chemistry, 2007
• Investigation of lipophilicity of anticancer‐active thioquinoline derivatives
  Biomedical Chromatography, 2006
• Relationships between structure and high-throughput screening permeability of diverse drugs with artificial membranes: Application to prediction of Caco-2 cell permeability
  Bioorganic & Medicinal Chemistry, 2005
• Caco-2 permeability of weakly basic drugs predicted with the Double-Sink PAMPA method
  European Journal of Pharmaceutical Sciences, 2005
• PAMPA—a drug absorption in vitro model
  European Journal of Pharmaceutical Sciences, 2004
• Prediction of human intestinal permeability using artificial membrane permeability
  International Journal of Pharmaceutics, 2003
• A comparative study of artificial membrane permeability assay for high throughput profiling of drug absorption potential
  European Journal of Medicinal Chemistry, 2002
• Physicochemical High Throughput Screening: Parallel Artificial Membrane Permeation Assay in the Description of Passive Absorption Processes
  Journal of Medicinal Chemistry, 1998