From DEL Selections to Validated Hits to Clinical Leads

This publication has 84 references indexed in Scilit:

• 5-Aryl-4-carboxamide-1,3-oxazoles: Potent and selective GSK-3 inhibitors
  Bioorganic & Medicinal Chemistry Letters, 2012
• Getting physical in drug discovery II: the impact of chromatographic hydrophobicity measurements and aromaticity
  Drug Discovery Today, 2011
• Small-molecule discovery from DNA-encoded chemical libraries
  Chemical Society Reviews, 2011
• Counting individual DNA molecules by the stochastic attachment of diverse labels
  Proceedings of the National Academy of Sciences, 2011
• Drug Discovery with DNA-Encoded Chemical Libraries
  Bioconjugate Chemistry, 2010
• Selecting chemicals: the emerging utility of DNA-encoded libraries
  Current Opinion in Chemical Biology, 2010
• Autotaxin--an LPA producing enzyme with diverse functions
  The Journal of Biochemistry, 2010
• Structural Basis for Acetylated Histone H4 Recognition by the Human BRD2 Bromodomain
  Journal of Biological Chemistry, 2010
• Discovery of TNF Inhibitors from a DNA-Encoded Chemical Library based on Diels-Alder Cycloaddition
  Chemistry & Biology, 2009
• Ligand configurational entropy and protein binding
  Proceedings of the National Academy of Sciences, 2007