One-pot imination / Arbuzov reaction of 4-aminobutanal derivatives: Synthesis of 2-phosphorylpyrrolidines and evaluation of anticancer activity
Authors:
- Andrey V. SmolobochkinASAndrey V. Smolobochkin
- Rakhymzhan A. TurmanovRTRakhymzhan A. Turmanov
- Almir S. GazizovAGAlmir S. Gazizov
- Alexandra D. VoloshinaAVAlexandra D. Voloshina
- Julia K. VoroninaJVJulia K. Voronina
- Anastasiia S. SapunovaASAnastasiia S. Sapunova
- Alexander R. BurilovABAlexander R. Burilov
- Michail A. PudovikMPMichail A. Pudovik
- 1 August 2020
- journal article
- research article
- Published by Elsevier in Tetrahedron
- Vol. 76 (33)
Abstract
No abstract availableKeywords
Funding Information
- Ministry of Education and Science of the Russian Federation
This publication has 39 references indexed in Scilit:
- Triflic acid-mediated phenylation of N-acylaminoalkyl diethylacetals and N-acyl-2-phenyl cyclic amidesOrganic & Biomolecular Chemistry, 2011
- Activity‐Based Probes for Monitoring Postproline Protease ActivityChemBioChem, 2009
- Facile synthesis of cyclic α-perfluoroalkyl-α-aminophosphonatesJournal of Fluorine Chemistry, 2009
- Development of Potent and Selective Phosphinic Peptide Inhibitors of Angiotensin-Converting Enzyme 2Journal of Medicinal Chemistry, 2008
- A Versatile Annulation Protocol toward Novel Constrained Phosphinic PeptidomimeticsThe Journal of Organic Chemistry, 2007
- Synthesis, kinetic evaluation, and utilization of a biotinylated dipeptide proline diphenyl phosphonate for the disclosure of dipeptidyl peptidase IV-like serine proteasesBiochemical and Biophysical Research Communications, 2006
- Dipeptide proline diphenyl phosphonates are potent, irreversible inhibitors of seprase (FAPα)Biochemical and Biophysical Research Communications, 2006
- Synthetic Methods for Azaheterocyclic Phosphonates and Their Biological ActivityChemical Reviews, 2004
- LevetiracetamCNS Drugs, 1997
- Synthesis and biological activity of carboxylic acid replacement analogs of the potent angiotensin converting enzyme inhibitor 5(S)-benzamido-4-oxo-6-phenylhexanoyl-L-prolineJournal of Medicinal Chemistry, 1985