Approaches to improve metabolic stability of a statine-based GRP receptor antagonist
Authors:
- 1 February 2017
- journal article
- Published by Elsevier in Nuclear Medicine and Biology
- Vol. 45, 22-29
Abstract
No abstract availableKeywords
This publication has 29 references indexed in Scilit:
- GRP Receptor Imaging of Prostate Cancer Using [99mTc]Demobesin 4: a First-in-Man StudyMolecular Imaging and Biology, 2014
- In Vitro and In Vivo Evaluation of a 18F-Labeled High Affinity NOTA Conjugated Bombesin Antagonist as a PET Ligand for GRPR-Targeted Tumor ImagingPLOS ONE, 2013
- Gastrin Releasing Peptide Receptor-Directed Radioligands Based on a Bombesin Antagonist: Synthesis, 111In-Labeling, and Preclinical ProfileJournal of Medicinal Chemistry, 2013
- Nuclear Imaging Probes: from Bench to BedsideClinical Cancer Research, 2007
- Radiolabeled somatostatin receptor antagonists are preferable to agonists forin vivopeptide receptor targeting of tumorsProceedings of the National Academy of Sciences, 2006
- Gastrin-Releasing Peptide Receptors in Normal and Neoplastic Human Uterus: Involvement of Multiple Tissue CompartmentsThe Journal of Clinical Endocrinology & Metabolism, 2005
- Potent Bombesin-like Peptides for GRP-Receptor Targeting of Tumors with 99mTc: A Preclinical StudyJournal of Medicinal Chemistry, 2004
- Technetium-99m RP527, a GRP analogue for visualisation of GRP receptor-expressing malignancies: a feasibility studyEuropean Journal of Nuclear Medicine and Molecular Imaging, 2000
- The presence of receptors for bombesin/GRP and mRNA for three receptor subtypes in human ovarian epithelial cancersRegulatory Peptides, 2000
- Gastrin-Releasing Peptide Receptors in Non-Neoplastic and Neoplastic Human BreastThe American Journal of Pathology, 1999