Fluorescence-based assays for the assessment of drug interaction with the human transporters OATP1B1 and OATP1B3
- 1 October 2010
- journal article
- Published by Elsevier in Analytical Biochemistry
- Vol. 405 (1) , 50-58
Abstract
No abstract availableKeywords
Funding Information
- National Institutes of Health Small Business Innovation Research (R43GM086970)
This publication has 33 references indexed in Scilit:
- Evaluation of 4′,6-Diamidino-2-phenylindole as a Fluorescent Probe Substrate for Rapid Assays of the Functionality of Human Multidrug and Toxin Extrusion ProteinsDrug Metabolism and Disposition, 2010
- Development of a Cell-Based High-Throughput Assay to Screen for Inhibitors of Organic Anion Transporting Polypeptides 1B1 and 1B3Current Chemical Genomics, 2010
- Membrane transporters in drug developmentNature Reviews Drug Discovery, 2010
- Down-regulation of Na+/H+ Exchanger Regulatory Factor 1 Increases Expression and Function of Multidrug Resistance Protein 4Cancer Research, 2008
- The Human Multidrug Resistance Protein 4 (MRP4, ABCC4): Functional Analysis of a Highly Polymorphic GeneThe Journal of Pharmacology and Experimental Therapeutics, 2008
- Effect of pregnane X receptor ligands on transport mediated by human OATP1B1 and OATP1B3European Journal of Pharmacology, 2008
- Species Difference in the Inhibitory Effect of Nonsteroidal Anti-Inflammatory Drugs on the Uptake of Methotrexate by Human Kidney SlicesThe Journal of Pharmacology and Experimental Therapeutics, 2007
- Synthesis and Fluorescence of N , N , N ‐Trimethyl‐2‐[methyl(7‐nitrobenzo[ c ][l,2,5]oxadiazol‐4‐yl) amino]ethanaminium Iodide, a pH‐Insensitive Reporter of Organic Cation TransportSynthetic Communications, 2006
- Can the pharmaceutical industry reduce attrition rates?Nature Reviews Drug Discovery, 2004
- A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening AssaysSLAS Discovery, 1999