Novel potent and selective αvβ3/αvβ5 integrin dual antagonists with reduced binding affinity for human serum albumin

This publication has 40 references indexed in Scilit:

• Non-peptidic αvβ3 antagonists containing indol-1-yl propionic acids
  Bioorganic & Medicinal Chemistry Letters, 2005
• Solid-phase synthesis of a small library of 3-phenylthio-3-nicotinyl propionic acid derivatives acting as antagonists of the integrin αVβ3
  Bioorganic & Medicinal Chemistry Letters, 2004
• Nonpeptide α_vβ₃ Antagonists. 8. In Vitro and in Vivo Evaluation of a Potent α_vβ₃ Antagonist for the Prevention and Treatment of Osteoporosis
  Journal of Medicinal Chemistry, 2003
• Non-Peptide αvβ3 antagonists. Part 6: Design and synthesis of αvβ3 antagonists containing a pyridone or pyrazinone central scaffold
  Bioorganic & Medicinal Chemistry Letters, 2003
• Phenylbutyrates as potent, orally bioavailable vitronectin receptor (integrin αvβ3) antagonists
  Bioorganic & Medicinal Chemistry Letters, 2003
• Integrins
  Cell, 2002
• Integrin αvβ3 antagonists promote tumor regression by inducing apoptosis of angiogenic blood vessels
  Cell, 1994
• Protein binding of quinolonecarboxylic acids. I. Cinoxacin, nalidixic acid and pipemidic acid.
  Chemical and Pharmaceutical Bulletin, 1989
• Complete amino acid sequence of human serum albumin
  FEBS Letters, 1975
• Amino acid sequence adjoining the lone tryptophan of human serum albumin. A binding site of the protein
  Biochemistry, 1970