A survey of core replacements in indole-based HIV-1 attachment inhibitors
Authors:
- 1 June 2019
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 29 (11) , 1423-1429
Abstract
No abstract availableKeywords
This publication has 47 references indexed in Scilit:
- In VitroAntiviral Characteristics of HIV-1 Attachment Inhibitor BMS-626529, the Active Component of the Prodrug BMS-663068Antimicrobial Agents and Chemotherapy, 2012
- Design, synthesis and SAR of thienopyridines as potent CHK1 inhibitorsBioorganic & Medicinal Chemistry Letters, 2010
- Discovery of a small molecule inhibitor through interference with the gp120–CD4 interactionBioorganic & Medicinal Chemistry Letters, 2009
- Heterobiaryl Human Immunodeficiency Virus Entry InhibitorsJournal of Medicinal Chemistry, 2009
- Inhibitors of HIV-1 attachment. Part 2: An initial survey of indole substitution patternsBioorganic & Medicinal Chemistry Letters, 2009
- Conformational Evaluation of Indol-3-yl-N-alkyl-glyoxalylamides and Indol-3-yl-N,N-dialkyl-glyoxalylamidesSpectroscopy Letters, 2009
- Conformation–activity relationship on novel 4-pyridylmethylthio derivatives with antiangiogenic activityBioorganic & Medicinal Chemistry Letters, 2008
- Konformation und Rotationsbarrieren substituierter GlyoxylsäureamideAdvanced Synthesis & Catalysis, 1997
- The Indol-2-ylglyoxylamide Moiety: A New Building Block for the Design and Self-Assembly of Hydrogen Bond NetworksJournal of the American Chemical Society, 1996
- Indazole and indoline as aromatic bioisosteres in the imidazole class of serotonin 5-HT3 receptor antagonistsBioorganic & Medicinal Chemistry Letters, 1992