A novel bivalent albumin binder for enhanced tumor retention of a fibroblast activation protein-targeted radioligand
- 27 November 2025
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Chemical Communications
- Vol. 61 (96) , 19072-19075
Abstract
A novel bivalent albumin binder composed of two molecules of Lys-4-( p -iodophenyl)butyric acid markedly enhanced tumor retention of a FAP-targeted radioligand, suggesting its promising potential as a versatile pharmacokinetic modifier of radioligands.Keywords
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Funding Information
- Japan Agency for Medical Research and Development (JP24ama221604)
- Japan Agency for Medical Research and Development (JP25ama221604)
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