Psilocin analogs. 1. Synthesis of 3‐[2‐(dialkylamino)ethyl] ‐and 3‐[2‐(cycloalkylamino)ethyl] indol‐4‐ols
Authors:
- 1 February 1977
- journal article
- research article
- Published by Wiley in Journal of Heterocyclic Chemistry
- Vol. 14 (1) , 71-74
Abstract
The synthesis of four dialkyl and three eyeloalkyl analogs of psilocin (4, R ‐ CH3), a hallucinogenic principle found in certain fungi, is described. The synthetic route involves four transformations starting with 6,7‐dihydroindol‐4(5H)one: (1).Keywords
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