Chiral azole derivatives. Part 5: Synthesis of enantiomerically pure 1-[α-(benzofuran-2-yl)arylmethyl]-1H-1,2,4-triazoles, antifungal and antiaromatase agents
Authors:
- Flavia MessinaFMFlavia Messina
- Maurizio BottaMBMaurizio Botta
- Federico CorelliFCFederico Corelli
- Antonella PaladinoAPAntonella Paladino
- 1 December 2000
- journal article
- Published by Elsevier in Tetrahedron: Asymmetry
- Vol. 11 (24) , 4895-4901
Abstract
No abstract availableThis publication has 8 references indexed in Scilit:
- Chiral Azole Derivatives. 4.1 Enantiomers of Bifonazole and Related Antifungal Agents: Synthesis, Configuration Assignment, and Biological EvaluationThe Journal of Organic Chemistry, 2000
- Stereoselective synthesis of α-aryl-2-benzofuranmethanamines and α-aryl-1H-indole-2-methanamines through palladium-mediated annulation of chiral α-arylpropargylaminesTetrahedron: Asymmetry, 2000
- Chiral azole derivatives, 3. Synthesis of the enantiomers of the potent aromatase inhibitor 1-[2-benzofuranyl(4-chlorophenyl)methyl]-1H-imidazoleTetrahedron Letters, 1999
- Resolution of (±)-1-Aryl-2-propynylamines via Acyltransfer Catalyzed byCandida antarcticaLipaseThe Journal of Organic Chemistry, 1999
- N‐Alkyloxycarbonyl‐3‐aryloxaziridines: Their Preparation, Structure, and Utilization As Electrophilic Amination ReagentsChemistry – A European Journal, 1997
- Molecular Modeling of Azole Antifungal Agents Active against Candida albicans. 1. A Comparative Molecular Field Analysis StudyJournal of Medicinal Chemistry, 1996
- Substituted 1-[(benzofuran-2-YL)-phenylmethyl]-imidazoles as potent inhibitors of aromatase in vitro and in female rats in vivoThe Journal of Steroid Biochemistry and Molecular Biology, 1993
- Notes - Triazines. XVI. A New Synthesis for 1,2,4-TriazolesThe Journal of Organic Chemistry, 1956