Practical Synthesis of FEt-penta-cyclofenil and Its Derivatives for Potential PET Imaging
Authors:
- 15 October 2010
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 40 (22) , 3322-3331
Abstract
Generally, FEt-penta-cyclofenil and its derivatives have greater relative binding affinity to estradiol receptors than estradiol. (4-Fluoroethoxyphenyl)–(4′-hydroxyphenyl) methylenecyclopentane and its derivatives were synthesized for potential radioactive image agents, and their structures were characterized by ultraviolet, infrared, 1H NMR, 19F NMR, and high-resolution mass spectrometry.Keywords
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