One-pot two-step radioiodination based on copper-mediated iododeboronation and azide–alkyne cycloaddition reaction
- 18 December 2023
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Chemical Communications
- Vol. 60 (6) , 714-717
Abstract
Copper-mediated one-pot two-step radioiodination proceeds under mild conditions. Furthermore, this methodology operates with continuous incorporation of reagents into the reaction system and a single-step purification.Keywords
Funding Information
- Japan Society for the Promotion of Science (22H02928, JP17K10377, JP17K19670)
- Ministry of Education, Culture, Sports, Science and Technology
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