Multicomponent one-pot synthesis of (dihydro-1H-benzo[d]imidazole) phosphonate
- 9 April 2019
- journal article
- research article
- Published by Taylor & Francis in Phosphorus, Sulfur, and Silicon and the Related Elements
- Vol. 194 (11) , 1062-1066
Abstract
We present a multicomponent reaction strategy to synthesize a (dihydro-1H-benzo[d]imidazole)phosphonate family of compounds, using benzimidazoles, diethyl chlorophosphate and aliphatic amines as starting reactants. Giving its simplicity, our procedure involves reaction times of only few hours and avoid the usage of any catalyst agent. All the newly synthesized compounds were characterized by Nuclear Magnetic Resonance spectroscopy (1H, 13C and 31P) and mass spectrometry by the DART method.Keywords
Funding Information
- Secretariat for Instituto Politecnico Nacional (20161237)
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